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Pazopanib (100 mg/kg/day free base equivalent)
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这是个已经在美国上市的老药了,能下载到正式药物使用说明书英文版。 2 w$ ]( f; T6 y6 _5 y" G搜索了一下,原料一大堆。8 A5 [: [' z" M
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对不起!100mg/kg是用于移植瘤的,我弄错了。9 a! I2 j' g! B8 z
7 e Y: j5 H Z% q" w3 l4 G9 I以下是正版说明书的推荐用量。/ b1 v& o$ |" [/ h# Q3 r) f
' q0 g$ k1 Y* w0 m% [--------------------- DOSAGE AND ADMINISTRATION ---------------- : }# [: r* h$ b) [* 800 mg orally once daily without food (at least 1 hour before or 2 hours after a meal). (2.1) / {5 g$ s$ s& Y' u J7 _4 h7 d
* Baseline moderate hepatic impairment – 200 mg orally once daily. Not recommended in patients with severe hepatic impairment. (2.2) & P1 `0 C+ u4 T/ L+ l' j& M---------------------DOSAGE FORMS AND STRENGTHS --------------" u5 e0 ~: c" n' t' T# t1 D2 t
200 mg tablets. (3) ; p8 W l( o/ {# \2 o
-------------------------------CONTRAINDICATIONS------------------------