平安! 发表于 2011-11-9 19:57 + D( n) }: }' [+ }% L
Pazopanib (100 mg/kg/day free base equivalent)
0 v4 @+ R+ ^4 F- G0 m% L- }3 D: a 这是个已经在美国上市的老药了,能下载到正式药物使用说明书英文版。( ^, [0 p4 E, S( [" K
搜索了一下,原料一大堆。! O& F9 L. Z2 s4 V& g4 s/ o
) r8 J$ F1 m" q1 m对不起!100mg/kg是用于移植瘤的,我弄错了。2 U3 R6 h; h/ D* j, f. |4 [0 ?
1 T" l$ Z* K3 K" Z5 H' z) b$ a以下是正版说明书的推荐用量。
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/ Z! h5 e0 R; ~, _" K) `8 {+ I--------------------- DOSAGE AND ADMINISTRATION ----------------; ^6 _ s. x3 r$ N( p3 y
* 800 mg orally once daily without food (at least 1 hour before or 2 hours after a meal). (2.1)
/ p/ L, q7 ~. s8 d) d! Y' W* Baseline moderate hepatic impairment – 200 mg orally once daily. Not recommended in patients with severe hepatic impairment. (2.2)
/ ]* ?1 n9 N7 x! }---------------------DOSAGE FORMS AND STRENGTHS --------------
' o, o3 Q1 z p" Q+ ^' {2 e200 mg tablets. (3)
/ Q: l% e: V7 y9 l3 T" s-------------------------------CONTRAINDICATIONS------------------------ |