平安! 发表于 2011-11-9 19:57 0 f9 S" x4 c) w
Pazopanib (100 mg/kg/day free base equivalent)
4 C4 ]' P. Z% Y7 P( D( z7 E 这是个已经在美国上市的老药了,能下载到正式药物使用说明书英文版。1 g+ q8 n+ i8 A4 Y, M l# F8 y7 w/ Q7 Z
搜索了一下,原料一大堆。4 W! c2 {- Z7 \4 O: W5 z" I* Z: `" s
! k& J. d! M: k+ \对不起!100mg/kg是用于移植瘤的,我弄错了。
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以下是正版说明书的推荐用量。! i4 Y5 N) ^3 e" ~* p2 L
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--------------------- DOSAGE AND ADMINISTRATION ----------------$ G$ J0 o! M9 q8 q7 f5 q0 {
* 800 mg orally once daily without food (at least 1 hour before or 2 hours after a meal). (2.1) - M5 z' a6 F3 W& X8 q
* Baseline moderate hepatic impairment – 200 mg orally once daily. Not recommended in patients with severe hepatic impairment. (2.2)
) @8 ^" c* `4 u" t, [' m3 e---------------------DOSAGE FORMS AND STRENGTHS --------------
( _& f5 {5 [ {* |200 mg tablets. (3) 8 H7 ?9 V; L4 `
-------------------------------CONTRAINDICATIONS------------------------ |