平安! 发表于 2011-11-9 19:57 & m, ^1 ]8 V0 M" ]$ ?% ]* \* N
Pazopanib (100 mg/kg/day free base equivalent)
5 H7 i( z; m. m* O% r: f% K# ? 这是个已经在美国上市的老药了,能下载到正式药物使用说明书英文版。; q# k2 d) W9 m$ u
搜索了一下,原料一大堆。- f" X/ B B- G* D+ @
! u) p7 b4 G& T# O6 }1 ?' F: v对不起!100mg/kg是用于移植瘤的,我弄错了。8 B1 S' Y0 P' O5 d. n6 H( p
" T3 }5 C5 A+ E+ n" h以下是正版说明书的推荐用量。5 ?+ n# Q! a: R1 r
/ ^/ ?2 l4 ~ V( L. I' N" b
--------------------- DOSAGE AND ADMINISTRATION ----------------
$ M' H# k, S7 G% m' _" }; I) \6 b' N% C* 800 mg orally once daily without food (at least 1 hour before or 2 hours after a meal). (2.1)
, q5 \" i$ B% c z. U7 ~. R: s" D* Baseline moderate hepatic impairment – 200 mg orally once daily. Not recommended in patients with severe hepatic impairment. (2.2)
8 J1 g% @/ ?# ?( [9 N$ B---------------------DOSAGE FORMS AND STRENGTHS --------------6 ] a- H% m. w" e" X/ C
200 mg tablets. (3) # F1 E3 L) l. Y' [
-------------------------------CONTRAINDICATIONS------------------------ |