平安! 发表于 2011-11-9 19:57
' N/ I# c u5 N2 NPazopanib (100 mg/kg/day free base equivalent)
; `6 m+ b: ~# ?% \8 {% d 这是个已经在美国上市的老药了,能下载到正式药物使用说明书英文版。! V$ y" e F1 V. o8 u' H f7 F8 ` O# N
搜索了一下,原料一大堆。0 M6 h8 U; p! A# [
$ i1 G" c6 @' w+ z! d. w对不起!100mg/kg是用于移植瘤的,我弄错了。# U. e4 v% E/ G3 @( ?
% v! l2 o' U @$ @- T" r以下是正版说明书的推荐用量。- ^* [7 o: I4 `) u0 }3 t
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--------------------- DOSAGE AND ADMINISTRATION ----------------6 v5 H9 B2 b" g5 I3 d) \7 l
* 800 mg orally once daily without food (at least 1 hour before or 2 hours after a meal). (2.1) 3 P' G P8 H9 _7 v1 x3 J, u& _0 c* k
* Baseline moderate hepatic impairment – 200 mg orally once daily. Not recommended in patients with severe hepatic impairment. (2.2)
R$ P% A/ }( S% u* o---------------------DOSAGE FORMS AND STRENGTHS --------------% v4 k |0 _- e" }
200 mg tablets. (3)
/ P, I c. I0 D Y6 W-------------------------------CONTRAINDICATIONS------------------------ |