平安! 发表于 2011-11-9 19:57
7 Q5 } z1 Z+ fPazopanib (100 mg/kg/day free base equivalent)
u. G' \& i6 L+ r) `2 i 这是个已经在美国上市的老药了,能下载到正式药物使用说明书英文版。
+ i; i, H* {3 ]$ ]搜索了一下,原料一大堆。
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0 g) C' a8 h+ d. {: J7 `+ W( i对不起!100mg/kg是用于移植瘤的,我弄错了。
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以下是正版说明书的推荐用量。4 i6 q1 X8 t- o9 K }
) U7 s5 _ v3 I7 w; H! {% p; [. u--------------------- DOSAGE AND ADMINISTRATION ----------------0 G8 ]% P1 { F* l' F( [% C
* 800 mg orally once daily without food (at least 1 hour before or 2 hours after a meal). (2.1)
' ^0 w+ A0 X& ?/ i [/ P7 ~* Baseline moderate hepatic impairment – 200 mg orally once daily. Not recommended in patients with severe hepatic impairment. (2.2) , z5 k6 `$ v, N# c- B
---------------------DOSAGE FORMS AND STRENGTHS --------------
, y* |" z% e" T( x0 p; Y200 mg tablets. (3) " \- J1 W- ~8 G$ v1 `( C6 }7 L
-------------------------------CONTRAINDICATIONS------------------------ |